Pharmacology/Part 10/10.2 Toxicology

10.2 Toxicology & Antidotes

Toxicology addresses poisoning, overdose management, and antidote therapy. Recognizing toxidromes and knowing specific antidotes can be life-saving.

Common Antidotes

ToxinAntidoteMechanism
AcetaminophenN-acetylcysteineReplenishes glutathione; prevents NAPQI toxicity
OpioidsNaloxoneฮผ-opioid receptor antagonist
BenzodiazepinesFlumazenilGABA-A receptor antagonist (caution: seizures)
WarfarinVitamin K, FFP, PCCReplenish clotting factors
HeparinProtamine sulfateBinds and neutralizes heparin
AnticholinergicsPhysostigmineAcetylcholinesterase inhibitor (crosses BBB)
OrganophosphatesAtropine + pralidoximeBlocks muscarinic effects; reactivates AChE
ฮฒ-blockers, CCBsGlucagon, calcium, insulinInotropic support, overcome blockade
DigoxinDigoxin-specific FabBinds and inactivates digoxin
IronDeferoxamineChelates free iron
LeadEDTA, succimer, dimercaprolChelation therapy
CyanideHydroxycobalamin, sodium thiosulfateBinds cyanide; provides sulfur for detox
Methanol, ethylene glycolFomepizole, ethanolInhibit alcohol dehydrogenase