Part 2: DNA Structure and Chemistry

The Blueprint of Life

DNA (deoxyribonucleic acid) is the molecular basis of heredityβ€”a polymer of extraordinary elegance that encodes the instructions for building and operating all known living organisms. Understanding its structure reveals how genetic information is stored, replicated, and transmitted across generations.

This section explores DNA from its basic chemical building blocks to its complex three-dimensional organization, covering the fundamental principles that make DNA uniquely suited to serve as the universal information molecule of life.

Historical Discovery

1869

Friedrich Miescher

Isolated "nuclein" from white blood cells in pus-soaked bandages, marking the first identification of DNA as a distinct substance.

1928

Frederick Griffith

Discovered bacterial transformation, demonstrating that genetic material could be transferred between organisms.

1944

Avery, MacLeod, McCarty

Proved that DNA (not protein) was the "transforming principle" and the carrier of genetic information.

1950

Erwin Chargaff

Discovered base pairing rules: A=T and G=C in equal proportions (Chargaff's rules).

1952

Rosalind Franklin

Produced Photo 51, the critical X-ray diffraction image showing DNA's helical structure.

1953

Watson & Crick

Proposed the double helix model, winning the 1962 Nobel Prize. Their famous paper in Nature began: "We wish to suggest a structure for the salt of deoxyribose nucleic acid (D.N.A.)."

Chapter Topics

DNA Chemical Components

DNA is a polymer composed of repeating units called nucleotides. Each nucleotide consists of three components:

1. Nitrogenous Base

The information-carrying component

Purines: Adenine (A), Guanine (G)

Pyrimidines: Cytosine (C), Thymine (T)

2. Deoxyribose Sugar

5-carbon pentose sugar

β€’ Missing 2'-OH group

β€’ More stable than ribose

β€’ Connects base to backbone

3. Phosphate Group

Links nucleotides together

β€’ Creates 5'β†’3' polarity

β€’ Negative charge

β€’ Phosphodiester bonds

The Phosphodiester Bond

Nucleotides are linked via phosphodiester bonds between the 5' phosphate of one nucleotide and the 3' hydroxyl of the next. This creates the sugar-phosphate backbone with inherent directionality (5'β†’3'), which is crucial for replication and transcription.

The Four DNA Bases

Purines (Two-Ring Structure)

Adenine (A)

6-aminopurine

  • β€’ Pairs with Thymine (2 H-bonds)
  • β€’ Amino group at C6 position
  • β€’ Found in ATP, NAD+, FAD

Guanine (G)

2-amino-6-oxopurine

  • β€’ Pairs with Cytosine (3 H-bonds)
  • β€’ Amino at C2, carbonyl at C6
  • β€’ Found in GTP, cGMP

Pyrimidines (One-Ring Structure)

Cytosine (C)

4-amino-2-oxopyrimidine

  • β€’ Pairs with Guanine (3 H-bonds)
  • β€’ Can be methylated (5-mC)
  • β€’ Prone to deamination β†’ Uracil

Thymine (T)

5-methyl-2,4-dioxopyrimidine

  • β€’ Pairs with Adenine (2 H-bonds)
  • β€’ Methylated C5 (vs. Uracil in RNA)
  • β€’ DNA-specific base

DNA Structure Overview

Key Dimensions (B-DNA)

Helix diameter2.0 nm (20 Γ…)
Rise per base pair0.34 nm (3.4 Γ…)
Base pairs per turn10.5
Helical pitch3.4 nm (34 Γ…)
Major groove width~22 Γ…
Minor groove width~12 Γ…

Base Pairing Rules

A═══ 2 H-bonds ═══T

Adenine-Thymine pair

G═══ 3 H-bonds ═══C

Guanine-Cytosine pair

Chargaff's Rules:

β€’ [A] = [T] and [G] = [C]

β€’ [Purines] = [Pyrimidines]

β€’ A+T/G+C ratio varies by species

Watson-Crick Base Pairing

The specific base pairing (A-T and G-C) is determined by the geometry of hydrogen bond donors and acceptors on the bases. A purine always pairs with a pyrimidine, maintaining the constant helix diameter. The three hydrogen bonds in G-C pairs make them stronger than A-T pairs, affecting DNA melting temperature and stability.

Forces Stabilizing DNA Structure

1. Hydrogen Bonds

Between complementary bases (A-T: 2 bonds, G-C: 3 bonds). Each bond contributes ~2-3 kcal/mol. While individually weak, the cumulative effect of millions of base pairs provides significant stability.

2. Base Stacking (Ο€-Ο€ Interactions)

The primary stabilizing force. Aromatic rings of adjacent bases stack atop each other, creating van der Waals interactions and hydrophobic effects. Contributes more to stability than hydrogen bonding. Each stack contributes ~5-10 kcal/mol.

3. Hydrophobic Effect

The hydrophobic bases are buried in the interior of the helix, away from water. The hydrophilic sugar-phosphate backbone faces the aqueous environment. This arrangement is thermodynamically favorable.

4. Ionic Interactions

Cations (Mg²⁺, K⁺, Na⁺, polyamines) neutralize the negative charges of the phosphate backbone, reducing electrostatic repulsion between the two strands. DNA is a polyanion with one negative charge per nucleotide.

DNA Conformational Forms

PropertyA-DNAB-DNAZ-DNA
Helix senseRight-handedRight-handedLeft-handed
Diameter26 Γ…20 Γ…18 Γ…
Rise per bp2.6 Γ…3.4 Γ…3.7 Γ…
Base pairs per turn1110.512
Helical pitch28 Γ…34 Γ…45 Γ…
Major grooveNarrow, deepWide, deepFlat
Minor grooveWide, shallowNarrow, deepNarrow, deep
ConditionsLow humidity, RNA-DNAPhysiologicalHigh salt, GC-rich

A-DNA

Found in dsRNA and RNA-DNA hybrids. Compact, dehydrated form.

B-DNA

Most common form in cells. Watson-Crick model represents B-DNA.

Z-DNA

Left-handed helix. May regulate transcription at promoter regions.

DNA Melting and Stability

DNA melting (denaturation) is the separation of the two strands when heated. The melting temperature (Tm)is the temperature at which 50% of the DNA is double-stranded.

Melting Temperature Calculation

For short oligonucleotides (<20 bp):

Tm = 4(G+C) + 2(A+T) Β°C

This rule works well for simple estimation of primer Tm

Factors Increasing Tm

  • β€’ Higher G-C content (3 H-bonds)
  • β€’ Longer DNA length
  • β€’ Higher salt concentration
  • β€’ Presence of Mg²⁺
  • β€’ Circular vs. linear DNA

Factors Decreasing Tm

  • β€’ Lower G-C content
  • β€’ Denaturants (urea, formamide)
  • β€’ Mismatches in sequence
  • β€’ Organic solvents
  • β€’ Low ionic strength

DNA Topology: Supercoiling

DNA in cells is not a simple linear moleculeβ€”it is supercoiled, meaning the double helix is itself twisted into a higher-order structure.

The Linking Number Equation

Lk = Tw + Wr
Lk

Linking Number

Number of times strands wrap

Tw

Twist

Helical winding of strands

Wr

Writhe

Superhelical coiling

Negative Supercoiling

Underwound DNA (Lk < Lkβ‚€). Common in most organisms. Facilitates strand separation for replication and transcription. Created by DNA gyrase.

Positive Supercoiling

Overwound DNA (Lk > Lkβ‚€). Found in some extremophiles. Generated ahead of replication forks. Removed by topoisomerases.

Chromatin: DNA Packaging

The human genome contains ~3.2 billion base pairs, stretching ~2 meters if fully extended. To fit into a nucleus ~6 ΞΌm in diameter, DNA must be compacted ~10,000-fold. This is achieved through hierarchical packaging into chromatin.

1

Nucleosome (11 nm fiber)

147 bp of DNA wrapped 1.65 turns around histone octamer (H2A, H2B, H3, H4 Γ— 2)

2

Chromatin Fiber (30 nm)

Nucleosomes fold into higher-order structure, stabilized by H1 linker histone

3

Chromatin Loops (300 nm)

30 nm fiber forms loops attached to protein scaffold

4

Metaphase Chromosome (1400 nm)

Maximum compaction during cell division; visible under light microscope

Compaction Ratio

Relaxed DNA β†’ Metaphase chromosome: ~10,000Γ— compaction
Interphase nucleus: ~1,000Γ— compaction (allows transcription)

Key Equations and Values

Molecular Weight of DNA

MW β‰ˆ n Γ— 330 Da (where n = number of nucleotides)

Average MW per nucleotide ~330 daltons

Length of DNA

Length (nm) = n Γ— 0.34 (where n = number of base pairs)

Each base pair rises 0.34 nm (3.4 Γ…) along the helix

Number of Helical Turns

Turns = n / 10.5 (for B-DNA)

B-DNA has 10.5 bp per turn

Human Genome Size

3.2 Γ— 10⁹ bp Γ— 0.34 nm/bp = 1.1 Γ— 10⁹ nm β‰ˆ 2 meters

Per diploid cell (23 chromosome pairs)

Learning Objectives

After completing Part 2, you should be able to:

  • βœ“Describe the chemical structure of nucleotides and nucleic acids
  • βœ“Explain Watson-Crick base pairing and Chargaff's rules
  • βœ“Compare different DNA conformations (A, B, Z forms)
  • βœ“Calculate DNA length, molecular weight, and helical turns
  • βœ“Identify forces that stabilize the double helix
  • βœ“Understand DNA topology and supercoiling
  • βœ“Explain the linking number equation (Lk = Tw + Wr)
  • βœ“Describe the role of topoisomerases
  • βœ“Outline chromatin organization and nucleosome structure
  • βœ“Calculate DNA melting temperature

Clinical Relevance

Topoisomerase Inhibitors

Anticancer drugs (doxorubicin, etoposide, topotecan) and antibiotics (ciprofloxacin) target topoisomerases, blocking DNA replication in rapidly dividing cells or bacteria.

DNA Repair Disorders

Defects in DNA structure recognition lead to diseases like Xeroderma Pigmentosum and Werner Syndrome. Understanding DNA chemistry is key to developing treatments.

Epigenetics

DNA methylation and histone modifications alter chromatin structure without changing the sequence, affecting gene expression in development and disease.

PCR and Diagnostics

Understanding DNA melting and annealing is essential for PCR primer design, used in genetic testing, pathogen detection, and forensics.